This is a list of currently marketed formulations of estradiol benzoate (EB) throughout the world. Both EB alone and combinations of EB with other medications are included. The brand name, manufacturers, and countries marketed are listed. Discontinued or no longer marketed formulations of EB are not listed. The formulations listed unless otherwise indicated are generally oil solutions for intramuscular injection.
Estradiol benzoate alone Agofollin Depot (BB Pharma; Czech Republic, Slovakia) [microcrystalline aqueous suspension for intramuscular injection] Benzo-Ginestryl (Sanofi-Aventis; Mexico) Estradiol Benzoate Astar (Astar; Taiwan) Estradiol Benzoate Tai Yu (Tai Yu; Taiwan) Estradiol Benzoato Pharma Arte (Pharma Arte; Paraguay) Estramon (CCPC / Hexal; Lithuania, Taiwan) Imegiol (Imeg; Paraguay) Oestradiol Benzoate March (March Pharma; Thailand) Yi Tai Li (Maidihai; China)
Veterinary Bomerol for Cattle (Bayer Australia Ltd Animal Health; Australia) Mesalin (Intervet; Poland)
Estradiol benzoate plus progestogens
Estradiol benzoate/progesterone Ciclotest Forte (Quimica Janvier; Paraguay) Ciclovulan Forte (Farmical; Paraguay) Cumorit Forte (Taiwan Hemeilong; Taiwan) Damax (Offenbach; Mexico) Dispert GEN Fuerte (Dispert; Uruguay) Duogynon (CCM; Malaysia) Duoton (TP; Thailand) Duoton Fort T P (Thailand) Evacin (FA.PA.SA.; Paraguay) Feminal Forte (Sanifar; Paraguay) Gestrygen (Bruluart; Mexico) Lutes (Mochida Pharmaceutical; Japan) Lutofolone (Misr; Egypt) Lutoginestryl F (Sanofi-Aventis; Mexico) Menovis (Teofarma; Italy) Mestrolar (Paill; Belize, El Salvador, Guatemala, Honduras, Nicaragua) Metrigen Fuerte (Aspen Labs; Mexico) Nomestrol (Vijosa; Belize, El Salvador, Guatemala, Honduras, Nicaragua, Panama) Origeron (Kai Yuen; Hong Kong) Phenokinon-F (Vesco; Thailand) Primoson-F (Quimica Son's; Mexico) Pro-Estramon-S (Tai Yu; Taiwan) Prodiol (Gentle / Tai Yu; Taiwan) Proger-F (Streger; Mexico) Progestediol (Tai Yu; Taiwan) Progestradiol Forte (Lasca; Paraguay) Sinergon (Millet; Paraguay) Sinergon Forte (Millet Paraguay) Unitest Forte (Galeno; Paraguay) Vermagest (Vijosa; El Salvador, Honduras, Nicaragua)
Veterinary Component E-C (Elanco; South Africa) [implant] Component E-S (Elanco, South Africa) [implant] Synovex C (Zoetis; Canada, South Africa, United States) [implant] Synovex S (Zoetis; Australia, Canada, South Africa, United States) [implant]
Estradiol benzoate/progesterone/lidocaine Clinomin Forte (Medical Farmac; Paraguay) [microcrystalline aqueous suspension for intramuscular injection]
Estradiol benzoate/progesterone/tylosin
Veterinary Component E-C with Tylan (Elanco Animal Health; United States) [implant] Component E-S with Tylan (Elanco Animal Health; United States) [implant]
Estradiol benzoate/hydroxyprogesterone caproate Dos Dias N (Elea; Argentina) Primosiston (Bayer / BSP Bayer Schering Pharma; Argentina, Ecuador, Paraguay)
Estradiol benzoate plus androgens/anabolic steroids
Estradiol benzoate/testosterone propionate Bothermon (ASKA Seiyaku Asuka; Japan)
Veterinary Component E-H (Elanco; South Africa) [implant] Synovex H (Zoetis; Australia, Canada, South Africa, United States) [implant]
Estradiol benzoate/testosterone propionate/tylosin
Veterinary Component E-H (Elanco Animal Health; United States) [implant]
Estradiol benzoate/testosterone isobutyrate Folivirin (BB Pharma; Czech Republic) [microcrystalline aqueous suspension for intramuscular injection]
Estradiol benzoate/trenbolone acetate
Veterinary Synovex Choice (Zoetis; Canada, United States) [implant] Synovex One (Zoetis; United States) [implant] Synovex Plus (Zoetis; Canada, South Africa, United States) [implant] Synovex with Trenbolone Acetate (Zoetis; Australia) [implant]
Estradiol benzoate plus estrogens and androgens/anabolic steroids
Estradiol benzoate/estradiol phenylpropionate/testosterone propionate/testosterone phenylpropionate/testosterone isocaproate Estandron P (Organon; Brazil) Mixogen (Organon; India)
Estradiol benzoate plus miscellaneous agents
Estradiol benzoate/prednisolone/salicylic acid Alpicort E (Dr. August Wolff; Poland) [solution applied to the scalp] Alpicort F (Alcina / Dr. August Wolff / Remedia; Bulgaria, Croatia (Hrvatska), Czech Republic, Germany, Slovakia, Switzerland) [solution applied to the scalp] Alpicort Plus (Dr. August Wolff; Hungary) [solution applied to the scalp]
Estradiol benzoate/gentamicin/hydrocortisone/nystatin Cridermol Fem (EMPA; Paraguay) [vaginal cream] Ginabiot (Tecnofarma; Paraguay) [vaginal cream] Ginecovan (Farmical; Paraguay) [vaginal cream]
Discontinued estradiol benzoate formulations Estradiol benzoate/estradiol phenylpropionate (Dimenformon Prolongatum) Estradiol benzoate/estradiol dienanthate/testosterone enanthate benzilic acid hydrazone (Climacteron, Lactimex, Lactostat) Estradiol benzoate/estradiol valerate/hydroxyprogesterone caproate (Sin-Ol) Estradiol benzoate/monalazone (Malun 25) [vaginal tablet] Estradiol benzoate/progesterone (Sistocyclin) [microcrystalline aqueous suspension for intramuscular injection] Estradiol benzoate/progesterone/methandriol dipropionate (Progestandron) Estradiol benzoate/progesterone/testosterone propionate (Lukestra, Steratrin, Trihormonal, Trinestryl)
Veterinary Estradiol benzoate/estradiol enanthate/testosterone enanthate (Uni-Bol)
See also Estradiol benzoate § Available forms Estradiol benzoate § Availability List of combined sex-hormonal preparations
References